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Synthesis, structural characterisation, and preliminary evaluation of non-indolin-2-one-based angiogenesis inhibitors related to sunitinib (Sutent®)

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dc.contributor.authorSudta, Pichiten_AU
dc.contributor.authorKirk, Nicholasen_AU
dc.contributor.authorBezos, Annaen_AU
dc.contributor.authorGurlica, Anthonyen_AU
dc.contributor.authorMitchell, Rhysen_AU
dc.contributor.authorWeber, Thomasen_AU
dc.contributor.authorWillis, Anthonyen_AU
dc.contributor.authorPrabpai, Samranen_AU
dc.contributor.authorKongsaeree, Palangponen_AU
dc.contributor.authorSuksamrarn, Suniten_AU
dc.contributor.authorKelso, Michaelen_AU
dc.contributor.authorParish, Christopheren_AU
dc.date.accessioned2015-12-10T23:04:20Z
dc.date.issued2013
dc.date.updated2016-02-24T10:25:49Z
dc.description.abstractThe indolin-2-one fused-ring system and the 2,4-dimethylpyrrole unit represent key structural motifs in the anticancer drug sunitinib (Sutent®) and predecessor angiogenesis inhibitors that have undergone anticancer clinical trials (e.g. semaxanib, SU5416
dc.identifier.issn0004-9425
dc.identifier.urihttp://hdl.handle.net/1885/62321
dc.publisherCSIRO Publishing
dc.sourceAustralian Journal of Chemistry
dc.subjectKeywords: Angiogenesis inhibitors; Anti-angiogenic activity; Anticancer drug; Fused-ring system; In-vitro models; Intra-molecular hydrogen bonds; Structural characteristics; Structural motifs; Scaffolds; Hydrocarbons
dc.titleSynthesis, structural characterisation, and preliminary evaluation of non-indolin-2-one-based angiogenesis inhibitors related to sunitinib (Sutent®)
dc.typeJournal article
local.bibliographicCitation.issue8
local.bibliographicCitation.lastpage873
local.bibliographicCitation.startpage864
local.contributor.affiliationSudta, Pichit, Srinakharinwirot University
local.contributor.affiliationKirk, Nicholas, University of Wollongong
local.contributor.affiliationBezos, Anna, College of Medicine, Biology and Environment, ANU
local.contributor.affiliationGurlica, Anthony, University of Wollongong
local.contributor.affiliationMitchell, Rhys, University of Wollongong
local.contributor.affiliationWeber, Thomas, University of Wollongong
local.contributor.affiliationWillis, Anthony, College of Physical and Mathematical Sciences, ANU
local.contributor.affiliationPrabpai, Samran, Mahidol University
local.contributor.affiliationKongsaeree, Palangpon, Mahidol University
local.contributor.affiliationParish, Christopher, College of Medicine, Biology and Environment, ANU
local.contributor.affiliationSuksamrarn, Sunit, Srinakharinwirot University
local.contributor.affiliationKelso, Michael, University of Wollongong
local.contributor.authoruidBezos, Anna, u9107121
local.contributor.authoruidWillis, Anthony, u8512028
local.contributor.authoruidParish, Christopher, u6900322
local.description.embargo2037-12-31
local.description.notesImported from ARIES
local.identifier.absfor030606 - Structural Chemistry and Spectroscopy
local.identifier.absseo970103 - Expanding Knowledge in the Chemical Sciences
local.identifier.ariespublicationu4005981xPUB687
local.identifier.citationvolume66
local.identifier.doi10.1071/CH13219
local.identifier.scopusID2-s2.0-84882683064
local.identifier.thomsonID000323176800005
local.type.statusPublished Version

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