Faridoon, MrHussein, Waleed MVella, PeterUl Islam, NazarOllis, DavidSchenk, GerhardMcGeary, Ross Peter2015-12-100960-894Xhttp://hdl.handle.net/1885/60712The production of β-lactamases is an effective strategy by which pathogenic bacteria can develop resistance against β-lactam antibiotics. While inhibitors of serine-β-lactamases are widely used in combination therapy with β-lactam antibiotics, there aKeywords: 3 mercapto 1,2,4 triazole derivative; beta lactam antibiotic; beta lactamase inhibitor; captopril; imipenemase inhibitor; n acylated thiosemicarbazide; thiosemicarbazide derivative; triazole derivative; unclassified drug; article; controlled study; drug p 3-Mercapto-1,2,4-triazoles; Antibiotic resistance; Inhibition assays; Metallo-ß-lactamases; Thiosemicarbazides3-Mercapto-1,2,4-triazoles and N-acylated thiosemicarbazides as metallo-β-lactamase inhibitors201210.1016/j.bmcl.2011.10.1162016-02-24