Malins, Lara2019-07-261367-5931http://hdl.handle.net/1885/164731Transition-metal catalysis has unlocked new paradigms for the late-stage modification and cyclization of peptides by harnessing the innate reactivity of proteinogenic amino acids. The field is rapidly evolving, with recent advances encompassing three fundamental areas - heteroatom couplings, decarboxylative cross-couplings, and C-H functionalizations - which have markedly extended the scope of conventional peptide modification and bioconjugation strategies. The advances outlined herein facilitate access to high-value peptide targets with promising applications in materials science and drug discovery.application/pdfen-AU© 2018 Elsevier Ltdhttp://creativecommons.org/licenses/by-nc-nd/4.0/201810.1016/j.cbpa.2018.03.0192019-03-31CC-BY-NC-ND 4.0 license